F02110304 | Transport of potassium

Compound Dose Time Species Model Method Action Result Positive criterion Reference
Perhexiline decrease Positive 16
Perhexiline decrease Positive 16
Diazoxide EC50= 40mmol/L, saturation by 100mmol/L Primary Culture of Neonatal Rat Cardiac Ventricular Myocytes flow cytometry and quantitative image analysis of cells stained with fluorescent DC indicators. affect Positive 188
Pinacidil affect Positive 188
5-Hydroxydecanoate 500mmol/L Primary Culture of Neonatal Rat Cardiac Ventricular Myocytes flow cytometry and quantitative image analysis of cells stained with fluorescent DC indicators. affect Positive 188
Glibenclamide affect Positive 188
Glibenclamide K1/2 values 1-6 microM heart and liver mitochondria from rat affect Positive 190