Database
User
| Full Name | Fo subunits |
|---|---|
| Subcellular Location | Mitochondrion membrane Multi-pass membrane protein |
| Compound | Dose | Time | Species | Model | Method | Result | Positive criterion | Reference |
|---|---|---|---|---|---|---|---|---|
| N,N'-dicyclohexylcarbodiimide | 1 mol inhibitor/mol F0 | E. coli | membrane H+-translocation | Positive | maximal inhibition | 170 | ||
| woodward's reagent k | Positive | 170 | ||||||
| Mersalyl | 130 μM | bovine | heart MF0, proton conductivity | Positive | 70% inhibition | 170 | ||
| Oligomycin | 152 μg inhibitor/mg protein | E. coli | membrane vesicle, pH gradient formation | Positive | 170 | |||
| Oligomycin | 7.1 μg inhibitor/mg protein | C. asciculate | SMP-ATPase | Positive | IC50 | 170 | ||
| Oligomycin | 2.0-3.0 μg inhibitor/mg protein | S. cerevisiae | SMP-ATPase | Positive | IC50 | 170 | ||
| Oligomycin | 0.3 μM | human NCI-60 cell lines | F0F1-ATPase | Positive | IC50 | 170 | ||
| Oligomycin | 15 ng inhibitor/mg protein | N. crassa | SMP-ATPase | Positive | Ki | 170 | ||
| Oligomycin | 0.21 μM | bovine | heart MF0F1-ATPase | Positive | Ki | 170 | ||
| Oligomycin | 0.4 μg inhibitor/mg protein | bovine | heart SMP-ATPase | Positive | 95% inhibition | 170 | ||
| Oligomycin | 0.5 μg/ml | rat | liver SMP-ATPase | Positive | 75% inhibition | 170 | ||
| ossamycin | 46 μg of inhibitor/mg protein | E. coli | pH gradient formation by membrane vesicle | Positive | IC50 | 170 | ||
| ossamycin | 8 μM | human NCI-60 cell lines | F0F1-ATPase | Positive | IC50 | 170 | ||
| ossamycin | 1.3 μg of inhibitor/mg protein | S. cerevisiae | SMP-ATPase | Positive | IC50 | 170 | ||
| venturicidin B | Positive | 170 | ||||||
| Bedaquiline | Positive | 170 | ||||||
| NCCD | 0.65 nmol/mg protein | bovine | heart SMP-ATPase | Positive | IC50 | 170 | ||
| NCCD | 1 nmol NCCD/mg protein | bovine | heart SMP-ATPase | Positive | 85% inhibition | 170 | ||
| N,N'-dicyclohexylcarbodiimide | 0.2 μg of inhibitor/mg protein | S. cerevisiae | SMP-ATPase | Positive | IC50 | 170 | ||
| N,N'-dicyclohexylcarbodiimide | 1-5 μg of inhibitor/mg protein | T. pyriformis | SMP-ATPase | Positive | IC50 | 170 | ||
| N,N'-dicyclohexylcarbodiimide | 200 μMa in less than 5 min and at ∼40 μMa in 30 min | R. rubrum | F1-ATPase | Positive | 170 | |||
| N,N'-dicyclohexylcarbodiimide | 1.9 μg/mg protein | C. fasciculata | SMP-ATPase | Positive | IC50 | 170 | ||
| N,N'-dicyclohexylcarbodiimide | 1 mol DCCD/mol F1 | EF1-ATPase | Positive | 95% inhibition | 170 | |||
| N,N'-dicyclohexylcarbodiimide | 30 μM | membrane-bound EF0F1-ATPase | Positive | maximal 70-80% inhibition | 170 | |||
| N,N'-dicyclohexylcarbodiimide | 5 μM | C. thermoaceticum | membrane-bound F0F1-ATPase | Positive | 47% inhibition | 170 | ||
| N,N'-dicyclohexylcarbodiimide | 2 mol inhibitor bound/mol F1 | bovine | heart MF1-ATPase | Positive | 97% inhibition | 170 | ||
| N,N'-dicyclohexylcarbodiimide | 1 mol inhibitor/mol F0 | bovine | heart SMP-ATPase | Positive | maximal inhibition | 170 | ||
| N,N'-dicyclohexylcarbodiimide | 2 mol inhibitor/mol F0 | bovine | heart H+-translocation | Positive | maximal inhibition | 170 | ||