Compound	Dose	Time	Species	Model	Method	Result	Positive criterion	Reference
AZD7545						Positive		256
VER-246608						Positive		256
JX06						Positive		256
radicicol						Positive		256
Oxythiamine						Positive		249
Dichloroacetate						Positive	IC50	255
2-chloroproprionate						Positive		255
Nov3r						Positive		255
Pfz3						Positive		255
AZD7545						Positive	IC50	255
radicicol						Positive		255
Dicoumarol	19.42 μM			ovarian cancer cell line SKOV3		Positive	IC50	256

T080001. [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial (EC 2.7.11.2) (Pyruvate dehydrogenase kinase isoform 1) (PDH kinase 1)
T080002. [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial (EC 2.7.11.2) (Pyruvate dehydrogenase kinase isoform 2) (PDH kinase 2) (PDKII)
T080003. [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial (EC 2.7.11.2) (Pyruvate dehydrogenase kinase isoform 3)
T080004. [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial (EC 2.7.11.2) (Pyruvate dehydrogenase kinase isoform 4)

F020401. glycolysis
F0202. Pyruvate metabolism